Darzen condensation
Drazen Condensation
This is the chemical reaction of a ketone or aldehyde with an α-haloester in the presence of a base to form an α,β-epoxy ester, also called a "glycidic ester". This reaction is also known as the Darzens condensation or glycidic ester condensation. In 1904 Auguste Georges Darzens, an organic chemist discovered this reaction.
Reaction mechanism:
A strong base is used to form a carbanion from haloester. This carbanion is easily formed due to its resonance-stabilization. This acts as a nucleophilic and attacks
another carbonyl compound, forming a new carbon–carbon bond. These first two steps are similar to a base-catalyzed aldol reaction.
An epoxide is formed as a result of an intramolecular SN2 attack by the oxygen anion on carbon baring halide ,thus displacing the halide. This reaction is thus a condensation reaction as there is a net loss of HCl when the two reactant molecules join.
- Kinetic control vs thermodynamic control
- Selectivity (stereo, regio, chemo)
- Active methylene compounds
- Aldol Condensation
- Claisen condensation
- Cross Claisen Condensation
- Reformatsky Reaction
- Stobbes Condensation
- Darzen condensation
- Perkin condensation
- Wittig Reaction
- Nucleophilic Substitution Reactions
- SN Reactions I
- SN Reactions II
- SN Reactions III
- Nucleophilic Substitution Prime Reactions
- Neighbouring group participation
- Aromatic Electrophilic Substitution Reactions
- NAS Elimination Addition
- NAS Addition Elimination
- Aromatic Nucleophilic Reactions (diazonium salts)
- Elimination Reactions
- Reactive intermediates
- Chapters 23
- Department Chemistry
- Teacher
Dr. Syed Gohar Taqi Kazimi